TY - JOUR AU - Alonso, Dulce AU - Vázquez Villa, María Del Henar AU - Gamo, Ana M. AU - Martínez Esperón, Maria F. AU - Tortosa, Mariola AU - Viso, Alma AU - Fernández de la Pradilla, Roberto AU - Junquera González, María Elena AU - Aicart Sospedra, Emilio AU - Martín-Fontecha Corrales, María Del Mar AU - Benhamú Salama, Bellinda AU - López Rodríguez, María Luz AU - Ortega Gutiérrez, Silvia PY - 2010 DO - 10.1021/ml100053y SN - 1948-5875 UR - https://hdl.handle.net/20.500.14352/114435 T2 - ACS Medicinal Chemistry Letters AB - In this work, we report the design and synthesis of a set of fluorescent probes targeting the human 5-HT1A receptor (h5-HT1AR). Among the synthesized compounds, derivative 4 deserves special attention as being a high-affinity ligand (Ki = 2 nM) with... LA - eng M2 - 249 PB - ACS Publications KW - GPCR KW - Serotonin 5-HT1A receptor KW - Fluorescent probes KW - Receptor visualization TI - Development of fluorescent ligands for the human 5-HT1A receptor TY - journal article VL - 1 ER -