TY - JOUR AU - Ragusa, Giulio AU - Gómez Cañas, María AU - Morales, Paula AU - Pazos, María AU - Rodríguez Cueto, Carmen Aurora AU - Asproni, Battistina AU - Cichero, Elena AU - Fossa, Paola AU - Pinna, Gerard AU - Jagerovic, Nadine AU - Fernández Ruiz, José Javier AU - Murineddu, Gabriele PY - 2017 DO - 10.1016/j.ejmech.2017.01.002 SN - 0223-5234 UR - https://hdl.handle.net/20.500.14352/93394 T2 - European Journal Medicinal Chemistry AB - In the last few years, cannabinoid type-2 receptor (CB2R) selective ligands have shown a great potential as novel therapeutic drugs in several diseases. With the aim of discovering new selective cannabinoid ligands, a series of... LA - eng M2 - 398 PB - Elsevier KW - ADME model KW - CB(2) antagonism KW - Cannabinoid receptors KW - Docking studies KW - Scaffold hopping KW - Synthesis TI - New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data and molecular docking TY - journal article VL - 15 ER -