TY - JOUR AU - Vázquez Villa, María Del Henar AU - González Vera, Juan Antonio AU - Benhamú Salama, Bellinda AU - Viso, Alma AU - Fernandez de la Pradilla, Roberto AU - Junquera González, María Elena AU - Aicart Sospedra, Emilio AU - López Rodríguez, María Luz AU - Ortega Gutiérrez, Silvia PY - 2010 DO - 10.1021/jm1007177 SN - 0022-2623 UR - https://hdl.handle.net/20.500.14352/114528 T2 - Journal of Medicinal Chemistry AB - In this work we report the synthesis of a set of labeled ligands targeting the human 5-HT6 receptor (h5-HT6R). Among the synthesized compounds, fluorescent probe 10 (Ki = 175 nM and Φf = 0.21) and biotinylated derivative 15 (Ki = 90 nM) deserve... LA - eng M2 - 7095 PB - ACS Publications KW - Serotonin 5-HT6 receptor KW - GPCR KW - Molecular probes KW - Receptor visualization TI - Development of molecular probes for the human 5-HT6 receptor TY - journal article VL - 53 ER -